Description

Y4R agonist-2 is a Y4R agonist with a Ki of 0.033 nM.—–C53H81N19O10—-[1]Konieczny A, et al. N-Terminus to Arginine Side-Chain Cyclization of Linear Peptidic Neuropeptide Y Y4 Receptor Ligands Results in Picomolar Binding Constants. J Med Chem. 2021 Nov 8. –2757328-63-3–1144.33—-O=C([C@@H](NC(CC1)=O)CCCNC(N)=N)N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N)=O)CC2=CC=C(O)C=C2)=O)CCCNC(N)=N)=O)CC(C)C)=O)CCCNC(NC(NCCCCNC1=O)=O)=N)=O)CC3=CNC4=CC=CC=C34–Others–10 mM in DMSO–Others—-Others–Peptides