UFP-803 (TFA)-Get quote

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UFP-803 TFA is a potent urotensin-II receptor (UT) ligand. UFP-803 TFA has lower residual agonist activity, so it may be an important tool for the investigations on the role played by the UT system in physiology and pathology[1].—Neuroscience-Neuromodulation–C50H64N10O12S2.xC2HF3O2—-[1]Camarda V, et, al. In vitro and in vivo pharmacological characterization of the novel UT receptor ligand [Pen5,DTrp7,Dab8]urotensin II(4-11) (UFP-803). Comparative Study Br J Pharmacol. 2006 Jan; 147(1): 92-100.—-1061.23 (free acid)—-OC(C(F)(F)F)=O.O=C([C@@H](NC([C@H](C(C)(SSC[C@H](NC([C@@H](NC([C@@H](NC1=O)CCN)=O)CC2=CC=C(C=C2)O)=O)C(N[C@H](C(O)=O)C(C)C)=O)C)NC([C@@H](N)CC(O)=O)=O)=O)CC3=CC=CC=C3)N[C@@H]1CC4=CNC5=CC=CC=C45–Cardiovascular Disease–H2O–Urotensin Receptor—-GPCR/G Protein–Peptides