Description

(Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin is a potent vasopressin V1 receptor (VP V1R) antagonist. (Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin significantly decreases the mean arterial pressure (MAP) in rats[1].—–C54H76N14O11—-[1]Levi DI, et al. High dietary salt amplifies osmoresponsiveness in vasopressin-releasing neurons. Cell Rep. 2021 Mar 16;34(11):108866. –129520-65-6–1097.27—-CCOC(C=C1)=CC=C1C[C@@H](NC(CC2=CC=CC=C2)=O)C(N[C@@H](CC3=CC=CC=C3)C(N[C@@H](CCC(N)=O)C(N[C@@H](CC(N)=O)C(N[C@@H](CCCCN)C(N4[C@@H](CCC4)C(N[C@H](C(N)=O)CCCNC(N)=N)=O)=O)=O)=O)=O)=O–Cardiovascular Disease–10 mM in DMSO–Vasopressin Receptor–V1a Receptor –GPCR/G Protein–Peptides