[Orn5]-URP (TFA)-Get quote

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[Orn5]-URP TFA is a potent and selective pure antagonist of Urotensin-II receptor (UT), with an pEC50 of 7.24. [Orn5]-URP TFA displays no agonist activity[1][2].—Neuroscience-Neuromodulation–C48H62N10O10S2.xC2HF3O2—-[1]Diallo M, et, al. [Orn5]URP acts as a pure antagonist of urotensinergic receptors in rat cortical astrocytes. Peptides. 2008 May; 29(5): 813-9.|[2]David C, et, al. Structure-activity relationships and structural conformation of a novel urotensin II-related peptide. Peptides. 2004 Oct; 25(10): 1819-30.—-1003.20 (free acid)—-OC(C(F)(F)F)=O.O=C([C@@H](NC([C@H](CSSC[C@H](NC([C@@H](NC([C@@H](NC1=O)CCCN)=O)CC2=CC=C(C=C2)O)=O)C(N[C@H](C(O)=O)C(C)C)=O)NC([C@@H](N)C)=O)=O)CC3=CC=CC=C3)N[C@H]1CC4=CNC5=CC=CC=C45–Cardiovascular Disease–H2O–Urotensin Receptor—-GPCR/G Protein–Peptides