Description
[Orn5]-URP is a potent and selective pure antagonist of Urotensin-II receptor (UT), with an pEC50 of 7.24. [Orn5]-URP displays no agonist activity[1][2].—Neuroscience-Neuromodulation–C48H62N10O10S2—-[1]Diallo M, et, al. [Orn5]URP acts as a pure antagonist of urotensinergic receptors in rat cortical astrocytes. Peptides. 2008 May; 29(5): 813-9.|[2]David C, et, al. Structure-activity relationships and structural conformation of a novel urotensin II-related peptide. Peptides. 2004 Oct; 25(10): 1819-30.–782485-03-4–1003.20—-[ACFW-{Orn}-YCV (Disulfide bridge:Cys2-Cys7)]–Cardiovascular Disease–H2O–Urotensin Receptor—-GPCR/G Protein–Peptides




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