Neuropeptide SF(mouse,rat) (TFA)-Get quote

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Neuropeptide SF (mouse,rat) TFA is a potent neuropeptide FF receptor agonist with Ki values are 48.4 nM and 12.1 nM for NPFF1 and NPFF2, respectively. Neuropeptide SF TFA increases the amplitude of the sustained current of heterologously expressed acid sensing ion channel 3 (ASIC3) [1].—Neuroscience-Neuromodulation–C42H66F3N13O12—-[1]K Jhamandas, et al. Facilitation of spinal morphine analgesia in normal and morphine tolerant animals by neuropeptide SF and related peptides.Peptides. 2006 May;27(5):953-63.|[2]C Gouardères, et al. Quantitative autoradiographic distribution of NPFF1 neuropeptide FF receptor in the rat brain and comparison with NPFF2 receptor by using [125I]YVP and [(125I]EYF as selective radioligands. Neuroscience. 2002;115(2):349-61.|[3]Miklós Jászberényi, et al. The actions of neuropeptide SF on the hypothalamic-pituitary-adrenal axis and behavior in rats.Regul Pept. 2014 Jan 10;188:46-51.—-1002.05—-O=C(N)[C@H](CC1=CC=CC=C1)NC([C@H](CCCNC(N)=N)NC([C@H](CCC(N)=O)NC([C@H]2N(C([C@H](C)NC([C@H](C)NC([C@H](CC(C)C)NC([C@H](CO)N)=O)=O)=O)=O)CCC2)=O)=O)=O.OC(C(F)(F)F)=O–Neurological Disease–10 mM in DMSO–Neuropeptide Y Receptor—-GPCR/G Protein;Neuronal Signaling–Peptides