Description

(N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8) (E-2078), a stable Dynorphin A (1–8) (HY-P2159) analog, is a kappa opioid receptor (KOR) agonist[1].—Neuroscience-Neuromodulation–C50H81N15O9—-[1]Butelman ER, et al. Effects of E-2078, a stable dynorphin A(1-8) analog, on sedation and serum prolactin levels in rhesus monkeys. Psychopharmacology (Berl). 1999 Nov;147(1):73-80.–103613-84-9–1036.27—-CCNC([C@@H](CC(C)C)NC([C@H](CCCNC(N)=N)N(C)C([C@H](CCCNC(N)=N)NC([C@H](CC(C)C)NC([C@@H](NC(CNC(CNC([C@@H](NC)CC1=CC=C(C=C1)O)=O)=O)=O)CC2=CC=CC=C2)=O)=O)=O)=O)=O–Neurological Disease–H2O–Opioid Receptor–κ Opioid Receptor/KOR–GPCR/G Protein;Neuronal Signaling–Peptides