Description

GRK2i TFA is a GRK2 inhibitory polypeptide that specifically inhibits Gβγ activation of GRK2. GRK2i TFA corresponds to the Gβγ-binding domain and acts as a cellular Gβγ antagonist[1].–80°C, 2 years; -20°C, 1 year (Powder, sealed storage, away from moisture)—-C152H257F3N50O43S—-[1]Jorge A Sierra-Fonseca, et al. Nerve growth factor induces neurite outgrowth of PC12 cells by promoting Gβγ-microtubule interaction. BMC Neurosci. 2014 Dec 31;15:132.—-3598.10–98.41–O=C([C@@H](N)CC1=CNC2=CC=CC=C12)N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N3[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N4[C@H](C(N[C@H](C(N[C@H](C(O)=O)CO)=O)CCCNC(N)=N)=O)CCC4)=O)CCCCN)=O)CC(N)=O)=O)CCCCN)=O)CCSC)=O)CCCCN)=O)CCC3)=O)C(C)C)=O)CCCNC(N)=N)=O)CCC(N)=O)=O)C(C)C)=O)CC(C)C)=O)CCC(N)=O)=O)CCC(N)=O)=O)C)=O)CCC(O)=O)=O)CCCNC(N)=N)=O)CC5=CC=C(O)C=C5)=O)C)=O)CC(O)=O)=O)CCCNC(N)=N)=O)CC(C)C)=O)CCC(O)=O)=O)CCCCN)=O)CCCCN.OC(C(F)(F)F)=O–Others–H2O : 100 mg/mL (ultrasonic)–G Protein-coupled Receptor Kinase (GRK)—-GPCR/G Protein–Peptides